Synthesis, characterization and biological activity of fluorescently labeled bedaquiline analogues
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چکیده
منابع مشابه
synthesis and characterization of potentially biological active cyclometallated organoplatinum(ii) complexes
this work is presented in five parts. in the first part preparation of the starting complex [pt(c^n)cl(dmso)], 1, in which c^n = n(1),c(2?)-chelated, deprotonated 2-phenylpyridine, and dmso = dimethylsulfoxide, and its reaction with 1 equiv of the biphosphine ligands bis(diphenylphosphino)amine, dppa, or bis(diphenylphosphino)methane, dppm, to give the complex [pt(c^n)cl(dppa)], 2, or [pt(c^n)c...
15 صفحه اولNovel Linezolid like Analogues: Synthesis, Characterization and Biological Evaluation
The synthesis of 4-(substituted benzylidene)-2-(pyrazin-2-yl) oxazol-5(4H)-one was achieved in two steps, In first step, pyrazine-2-carboxamide dissolved in EtOH, 10% KOH solution with ClCH2COOH produced compound 2-(pyrazine-2-carboxamido) acetic acid (II) and in second step, compound (II) in (CH3CO)2O with aromatic aldehyde, and catalyst potassium ace...
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the synthesis of 4-(substituted benzylidene)-2-(pyrazin-2-yl) oxazol-5(4h)-one was achieved in two steps, in first step, pyrazine-2-carboxamide dissolved in etoh, 10% koh solution with clch2cooh produced compound 2-(pyrazine-2-carboxamido) acetic acid (ii) and in second step, compound (ii) in (ch3co)2o with aromatic aldehyde, and catalyst potassium acetate produced title compounds 4-(substitut...
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ژورنال
عنوان ژورنال: RSC Advances
سال: 2016
ISSN: 2046-2069
DOI: 10.1039/c6ra22693k